SR-14968

SR-14968 is a drug that acts as a biased agonist of the μ-opioid receptors, selectively activating the G-protein signaling pathway, as opposed to activation through β-arrestin 2. It is structurally and functionally similar to compounds such as brorphine and SR-17018.
Like morphine, SR-14968 exhibits pronounced antagonistic activity in vitro, but in in vivo animal studies it exhibits the properties of a typical opioid agonist at high dosages. Despite this, the drug retains a more favorable safety profile compared to opioids that do not have biased agonistic activity, such as fentanyl. Drugs in this class are considered promising analgesics with a reduced risk of overdose and addiction compared to traditional opioids.

Regulatory status: At the moment, SR-14968 is classified as a research substance and its use for medical purposes outside scientific institutions is not allowed. When conducting research and handling this substance, it is extremely important to comply with legal regulations and safety regulations in order to avoid its misuse.

Technical Information:

Product Name:  SR-14968

Synonyms: US10751335, Example 2

CAS: 2133455-40-8

IUPAC: 3-[1-[1-(4-bromophenyl)ethyl]piperidin-4-yl]-5,6-dichloro-1H-benzimidazol-2-one

Molecular Formula: C₂₀H₂₀BrCl₂N₃O

Molecular Weight:  469.2 g/mol

Purity:  98.0 % min.

Formulations: A solid

SMILES: CC(C1=CC=C(C=C1)Br)N2CCC(CC2)N3C4=CC(=C(C=C4NC3=O)Cl)Cl

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